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Synthesis and anthelmintic activity of a series of pyrazino[2,1-a][2]benzazepine derivatives


Journal of Medicinal Chemistry 32(9): 2058-2062
Synthesis and anthelmintic activity of a series of pyrazino[2,1-a][2]benzazepine derivatives
The synthesis and structure-activity relationships of a series of 1,2,3,4,6,7,8,12b-octahydropyrazinoenzazepine derivatives are described. Many of these compounds were active in vitro against Taenia crassiceps.


Accession: 001962409

PMID: 2769679



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