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Synthesis of antifungal imidazoles and triazoles

Annals of the New York Academy of Sciences 544: 12-31

Synthesis of antifungal imidazoles and triazoles

The syntheses of antifungal N-vinyl-imidazoles by the imidazole transfer reaction that resulted in the advent of croconazole (Pilzcin) and the syntheses of azolylpropanolones and diazolylpropanols having systemic antifungal activities are described.

Accession: 001962542

PMID: 3214063

DOI: 10.1111/j.1749-6632.1988.tb40386.x

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