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Preparation of highly hindered steroid esters application of some newer methods of esterification


, : Preparation of highly hindered steroid esters application of some newer methods of esterification. Steroids 34(7): 793-798

The scope and limitation of some recent acylation methods were investigated as applied to the preparation of steroidal esters of highly hindered acids. As representative steroids, 19-nor-17.alpha.-ethinyl testosterone (19-NET) and testosterone, and as representative acid, pivalic (trimethylacetic) acid were used. Potential anti-fertility uses are discussed.

Accession: 006173226

PMID: 538779

DOI: 10.1016/0039-128x(79)90091-6

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