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Synthesis and antiulcer activity of 2-amino-8H-indeno(1,2-d)thiazole derivatives


Yakugaku Zasshi 114(7): 523-532
Synthesis and antiulcer activity of 2-amino-8H-indeno(1,2-d)thiazole derivatives
A series of 8H-indeno(1,2-d)thiazoles containing various N-substituted amino groups at the 2 position were synthesized by the reaction of 2-bromo-indanones and N-substituted thioureas. Their anti-ulcerous activity was evaluated. Alkylamino derivatives have a more potent inhibitory behavior on ethanol-induced gastric ulcers compared with arylamino derivatives.


Accession: 009503984



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