Section 12
Chapter 11,093

Opioid peptide receptor studies. 15. Relative efficacy of 4- ( (N-allyl-3-methyl-4-piperidinyl) phenylamino) -N,N-diethylbenzamide and related compounds at the cloned human delta-opioid receptor

Xu, H.; Lu, Y.-Feng; Thomas, J., B.; Carroll, F.I.; Rice, K., C.; Rothman, R., B.

Synapse (New York) 40(4): 269-274


ISSN/ISBN: 0887-4476
Accession: 011092258

Previous data obtained from both binding and functional assays demonstrated that (-)-4-((N-allyl-3-methyl-4-piperidinyl)phenylamino)-N,N-diethylbenzamide ((-)-RTI5989-54) displays selective binding and full agonist activity relative to (+-)-RTI5989-54 for the delta opioid receptor.

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