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Structure-function relationship between analogues of the antibacterial peptide indolicidin. I. Synthesis and biological activity of analogues with increased amphipathicity and elevated net positive charge of the molecule

Structure-function relationship between analogues of the antibacterial peptide indolicidin. I. Synthesis and biological activity of analogues with increased amphipathicity and elevated net positive charge of the molecule

Bioorganicheskaia Khimiia 30(5): 458-465

ISSN/ISBN: 0132-3423

PMID: 15562965

DOI: 10.1023/b:rubi.0000043782.21640.c2

The antibacterial peptide indolicidin and a number of its analogues were obtained by solid phase synthesis. An optimized method of the synthesis using the Boc strategy was suggested.

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Accession: 012592211

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