Localization of the quinacrine noncompetitive inhibitor binding site on the open-channel conformation of the Torpedo acetylcholine receptor
Johnson, D.A.; Aryes, S.
Biophysical Journal 70(2 Part 2): A98
1996
ISSN/ISBN: 0006-3495
Accession: 032180988
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Related References
Johnson, D.A.; Ayres, S. 1996: Quinacrine noncompetitive inhibitor binding site localized on the Torpedo acetylcholine receptor in the open state Biochemistry 35(20): 6330-6336Arias, H.R.; Valenzuela, C.F.; Johnson, D.A. 1993: Transverse localization of the quinacrine binding site on the Torpedo acetylcholine receptor Journal of Biological Chemistry 268(9): 6348-6355
Pedersen, S.E.; Papineni, R.V. 1995: Interaction of d-tubocurarine analogs with the Torpedo nicotinic acetylcholine receptor. Methylation and stereoisomerization affect site-selective competitive binding and binding to the noncompetitive site Journal of Biological Chemistry 270(52): 31141-31150
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Gallagher, M.J.; Cohen, J.B. 1999: Identification of amino acids of the torpedo nicotinic acetylcholine receptor contributing to the binding site for the noncompetitive antagonist [(3)H]tetracaine Molecular Pharmacology 56(2): 300-307
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Pedersen, S.E.; Sharp, S.D.; Liu, W.S.hyong 1992: Structure of the noncompetitive antagonist-binding site of the Torpedo nicotinic acetylcholine receptor. (3H)meproadifen mustard reacts selectively with a-subunit Glu-262 Journal of Biological Chemistry 267: 489-499
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Tzartos, SJ.; Changeux, J-P. 1984: Lipid-dependent recovery of -bungarotoxin and monoclonal antibody binding to the purified -subunit from Torpedo marmorata acetylcholine receptor. Enhancement by noncompetitive channel blockers Journal of Biological Chemistry 259(18): 11512-11519