Solid-phase synthesis of head-to-tail cyclic peptides via lysine side-chain anchoring

Alsina, J.; Rabanal, F.; Giralt, E.; Albericio, F.

Tetrahedron Letters 35(51): 9633-9636

1994


ISSN/ISBN: 0040-4039
DOI: 10.1016/0040-4039(94)88531-1
Accession: 033428022

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Abstract
The N,N′-disuccinimidyl carbonate (DSC) has been successfully used for the efficient conversion of conventional hydroxymethyl resins into active carbonate resins, which are suitable for the incorporation of protected amino acids via an amino function, allowing the preparation of “head-to-tail” cyclic lysine containing peptides.