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Organocatalytic conjugate addition of malonates to alpha,beta-unsaturated aldehydes: asymmetric formal synthesis of (-)-paroxetine, chiral lactams, and lactones



Organocatalytic conjugate addition of malonates to alpha,beta-unsaturated aldehydes: asymmetric formal synthesis of (-)-paroxetine, chiral lactams, and lactones



Angewandte Chemie 45(26): 4305-4309




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Accession: 049819235

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PMID: 16646104

DOI: 10.1002/anie.200601025


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